Recent publications
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2-Alkyl substituted benzimidazoles as a new class of selective AT2 receptor ligands
Part of Bioorganic & Medicinal Chemistry, 2022.
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Nandrolone decanoate and testosterone undecanoate differently affect stress hormones, neurotransmitter systems, and general activity in the male rat
Part of Behavioural Brain Research, 2022.
DOI for Nandrolone decanoate and testosterone undecanoate differently affect stress hormones, neurotransmitter systems, and general activity in the male rat Download full text (pdf) of Nandrolone decanoate and testosterone undecanoate differently affect stress hormones, neurotransmitter systems, and general activity in the male rat
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Hydrogen Peroxide Induced Toxicity Is Reversed by the Macrocyclic IRAP-Inhibitor HA08 in Primary Hippocampal Cell Cultures
Part of Current Issues in Molecular Biology, p. 5000-5012, 2022.
DOI for Hydrogen Peroxide Induced Toxicity Is Reversed by the Macrocyclic IRAP-Inhibitor HA08 in Primary Hippocampal Cell Cultures Download full text (pdf) of Hydrogen Peroxide Induced Toxicity Is Reversed by the Macrocyclic IRAP-Inhibitor HA08 in Primary Hippocampal Cell Cultures
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The amino-terminal heptapeptide of the algesic substance P provides analgesic effect in relieving chronic neuropathic pain
Part of European Journal of Pharmacology, 2021.
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The effects of morphine, methadone, and fentanyl on mitochondria: A live cell imaging study
Part of Brain Research Bulletin, p. 126-134, 2021.
DOI for The effects of morphine, methadone, and fentanyl on mitochondria: A live cell imaging study
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Unilateral traumatic brain injury of the left and right hemisphere produces the left hindlimb response in rats
Part of Experimental Brain Research, p. 2221-2232, 2021.
DOI for Unilateral traumatic brain injury of the left and right hemisphere produces the left hindlimb response in rats Download full text (pdf) of Unilateral traumatic brain injury of the left and right hemisphere produces the left hindlimb response in rats
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Left-right side-specific neuropeptide mechanism mediates contralateral responses to a unilateral brain injury
Part of eNeuro, 2021.
DOI for Left-right side-specific neuropeptide mechanism mediates contralateral responses to a unilateral brain injury Download full text (pdf) of Left-right side-specific neuropeptide mechanism mediates contralateral responses to a unilateral brain injury
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Coordinated expression of the renin-angiotensin genes in the lumbar spinal cord: Lateralization and effects of unilateral brain injury
Part of European Journal of Neuroscience, p. 5560-5573, 2021.
DOI for Coordinated expression of the renin-angiotensin genes in the lumbar spinal cord: Lateralization and effects of unilateral brain injury Download full text (pdf) of Coordinated expression of the renin-angiotensin genes in the lumbar spinal cord: Lateralization and effects of unilateral brain injury
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Structurally different anabolic androgenic steroids reduce neurite outgrowth and neuronal viability in primary rat cortical cell cultures
Part of Journal of Steroid Biochemistry and Molecular Biology, 2021.
DOI for Structurally different anabolic androgenic steroids reduce neurite outgrowth and neuronal viability in primary rat cortical cell cultures Download full text (pdf) of Structurally different anabolic androgenic steroids reduce neurite outgrowth and neuronal viability in primary rat cortical cell cultures
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Assessing Cell Viability Effects of Opioids in Primary Cortical Cells from Rat.
Part of Methods in Molecular Biology, p. 171-180, 2021.
DOI for Assessing Cell Viability Effects of Opioids in Primary Cortical Cells from Rat.
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N-(Methyloxycarbonyl)thiophene sulfonamides as high affinity AT2 receptor ligands
Part of Bioorganic & Medicinal Chemistry, 2021.
DOI for N-(Methyloxycarbonyl)thiophene sulfonamides as high affinity AT2 receptor ligands
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Direct stimulation of angiotensin II type 2 receptor reduces nitric oxide production in lipopolysaccharide treated mouse macrophages
Part of European Journal of Pharmacology, 2020.
DOI for Direct stimulation of angiotensin II type 2 receptor reduces nitric oxide production in lipopolysaccharide treated mouse macrophages Download full text (pdf) of Direct stimulation of angiotensin II type 2 receptor reduces nitric oxide production in lipopolysaccharide treated mouse macrophages
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Anabolic androgenic steroids exert a selective remodeling of the plasma lipidome that mirrors the decrease of the de novo lipogenesis in the liver
Part of Metabolomics, 2020.
DOI for Anabolic androgenic steroids exert a selective remodeling of the plasma lipidome that mirrors the decrease of the de novo lipogenesis in the liver Download full text (pdf) of Anabolic androgenic steroids exert a selective remodeling of the plasma lipidome that mirrors the decrease of the de novo lipogenesis in the liver
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Growth hormone increases dendritic spine density in primary hippocampal cell cultures
Part of Growth Hormone & IGF Research, p. 42-47, 2020.
DOI for Growth hormone increases dendritic spine density in primary hippocampal cell cultures
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Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors
Part of ChemistryOpen, p. 325-337, 2020.
DOI for Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors Download full text (pdf) of Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors
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Macrocyclic Peptidomimetics as Inhibitors of Insulin-Regulated Aminopeptidase (IRAP)
Part of RSC Medicinal chemistry, p. 234-244, 2020.
DOI for Macrocyclic Peptidomimetics as Inhibitors of Insulin-Regulated Aminopeptidase (IRAP)
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Growing knowledge: How growth hormone improves learning
Part of Acta Physiologica, 2020.
DOI for Growing knowledge: How growth hormone improves learning
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Evolution of Angiotensin Peptides and Peptidomimetics as Angiotensin II Receptor Type 2 (AT2) Receptor Agonists
Part of Biomolecules, 2020.
DOI for Evolution of Angiotensin Peptides and Peptidomimetics as Angiotensin II Receptor Type 2 (AT2) Receptor Agonists Download full text (pdf) of Evolution of Angiotensin Peptides and Peptidomimetics as Angiotensin II Receptor Type 2 (AT2) Receptor Agonists
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Structural Basis of Inhibition of Insulin-Regulated Aminopeptidase by a Macrocyclic Peptidic Inhibitor
Part of ACS Medicinal Chemistry Letters, p. 1429-1434, 2020.
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Insulin-regulated aminopeptidase inhibitor-mediated increases in dendritic spine density are facilitated by glucose uptake
Part of Journal of Neurochemistry, p. 485-494, 2020.
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Ipsilesional versus contralesional postural deficits induced by unilateral brain trauma: a side reversal by opioid mechanism
Part of Brain Communications, 2020.
DOI for Ipsilesional versus contralesional postural deficits induced by unilateral brain trauma: a side reversal by opioid mechanism Download full text (pdf) of Ipsilesional versus contralesional postural deficits induced by unilateral brain trauma: a side reversal by opioid mechanism
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Toxic Impact of Anabolic Androgenic Steroids in Primary Rat Cortical Cell Cultures
Part of Neuroscience, p. 172-183, 2019.
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A Series of Analogues to the AT2R Prototype Antagonist C38 Allow Fine Tuning of the Previously Reported Antagonist Binding Mode
Part of ChemistryOpen, p. 114-125, 2019.
DOI for A Series of Analogues to the AT2R Prototype Antagonist C38 Allow Fine Tuning of the Previously Reported Antagonist Binding Mode Download full text (pdf) of A Series of Analogues to the AT2R Prototype Antagonist C38 Allow Fine Tuning of the Previously Reported Antagonist Binding Mode
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A convenient transesterification method for synthesis of AT2 receptor ligands with improved stability in human liver microsomes
Part of Bioorganic & Medicinal Chemistry Letters, p. 519-522, 2018.
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Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides
Part of ACS Omega, p. 4509-4521, 2018.
DOI for Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides Download full text (pdf) of Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides
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Chronic administration of morphine using mini-osmotic pumps affects spatial memory in the male rat
Part of Pharmacology, Biochemistry and Behavior, p. 1-8, 2018.
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An imidazole based H-Phe-Phe-NH2 peptidomimetic with anti-allodynic effect in spared nerve injury mice
Part of Bioorganic & Medicinal Chemistry Letters, p. 2446-2450, 2018.
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The Protective and Restorative Effects of Growth Hormone and Insulin-Like Growth Factor-1 on Methadone-Induced Toxicity In Vitro
Part of International Journal of Molecular Sciences, p. 1-16, 2018.
DOI for The Protective and Restorative Effects of Growth Hormone and Insulin-Like Growth Factor-1 on Methadone-Induced Toxicity In Vitro Download full text (pdf) of The Protective and Restorative Effects of Growth Hormone and Insulin-Like Growth Factor-1 on Methadone-Induced Toxicity In Vitro
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Impact of N-methylation of the substance P 1-7 amide on anti-allodynic effect in mice after peripheral administration
Part of European Journal of Pharmaceutical Sciences, p. 533-540, 2017.
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Importance of N-and C-terminal residues of substance P 1-7 for alleviating allodynia in mice after peripheral administration
Part of European Journal of Pharmaceutical Sciences, p. 345-351, 2017.
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The mRNA expression of insulin-like growth factor-1 (Igf1) is decreased in the rat frontal cortex following gamma-hydroxybutyrate (GHB) administration
Part of Neuroscience Letters, p. 15-20, 2017.
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Genetic susceptibility to postherniotomy pain. The influence of polymorphisms in the Mu opioid receptor, TNF-alpha, GRIK3, GCH1, BDNF and CACNA2D2 genes
Part of Scandinavian Journal of Pain, p. 1-6, 2016.
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Effects of growth hormone on brain function: new routes for the delivery of the hormone into the brain
Part of Amino Acids, p. 633-634, 2016.
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Identification of Drug-Like Inhibitors of Insulin-Regulated Aminopeptidase Through Small-Molecule Screening
Part of Assay and drug development technologies, p. 180-193, 2016.
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Aryl Sulfonamide Inhibitors of Insulin-Regulated Aminopeptidase Enhance Spine Density in Primary Hippocampal Neuron Cultures
Part of ACS Chemical Neuroscience, p. 1383-1392, 2016.
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[(35)S]GTPγS autoradiography for studies of opioid receptor functionality
Part of Methods in Molecular Biology, p. 169-176, 2015.
DOI for [(35)S]GTPγS autoradiography for studies of opioid receptor functionality
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Interconversion of Functional Activity by Minor Structural Alterations in Nonpeptide AT2 Receptor Ligands
Part of ACS Medicinal Chemistry Letters, p. 178-182, 2015.
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Small constrained SP1-7 analogues bind to a unique site and promote anti-allodynic effects following systemic injection in mice
Part of Neuroscience, p. 112-119, 2015.
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Inhibition of Insulin-Regulated Aminopeptidase (IRAP) by Arylsulfonamides
Part of ChemistryOpen, p. 256-263, 2014.
DOI for Inhibition of Insulin-Regulated Aminopeptidase (IRAP) by Arylsulfonamides
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Saralasin and Sarile Are AT2 Receptor Agonists
Part of ACS Medicinal Chemistry Letters, p. 1129-1132, 2014.
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Exploration and pharmacokinetic profiling of phenylalanine based carbamates as novel substance p 1-7 analogues
Part of ACS Medicinal Chemistry Letters, p. 1272-1277, 2014.
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Administration of growth hormone and nandrolone decanoate alters mRNA expression of the GABAB receptor subunits as well as of the GH receptor, IGF-1, and IGF-2 in rat brain.
Part of Growth Hormone & IGF Research, p. 60-66, 2014.
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Growth hormone reverses streptozotocin-induced cognitive impairments in male mice
Part of Behavioural Brain Research, p. 273-278, 2013.
DOI for Growth hormone reverses streptozotocin-induced cognitive impairments in male mice
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Application of in vitro [(35)S]GTPγ-S autoradiography in studies of growth hormone effects on opioid receptors in the male rat brain
Part of Brain Research Bulletin, p. 100-106, 2013.
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Constrained H-Phe-Phe-NH2 Analogues With High Affinity to the Substance P 1-7 Binding Site and With Improved Metabolic Stability and Cell Permeability
Part of Journal of Medicinal Chemistry, p. 4953-4965, 2013.